S83103 |
GSK-J2 |
源叶(MedMol) | ≥99% |
- 提示:详情请下载说明书。
- 产品描述: GSK-J2 is an isomer of GSK-J1 that does not have any specific activity. GSK-J1 is a potent inhibitor of H3K27me3/me2-demethylases JMJD3/KDM6B and UTX/KDM6A.
- 体外研究: GSK-J2 is an isomer of GSK-J1, and shows poor activity towards KDM6A and KDM6B, with IC50 of > 100 μM and 49 μM, respectively
- 参考文献:
1. Heinemann B, et al. Inhibition of demethylases by GSK-J1/J4. Nature. 2014 Oct 2;514(7520):E1-2
- 溶解性: soluble in DMSO
- 保存条件: -20℃
- 配置溶液浓度参考:
1mg 5mg 10mg 1 mM 2.568 ml 12.839 ml 25.677 ml 5 mM 0.514 ml 2.568 ml 5.135 ml 10 mM 0.257 ml 1.284 ml 2.568 ml 50 mM 0.051 ml 0.257 ml 0.514 ml
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本计算器可帮助您计算出特定溶液中溶质的质量、溶液浓度和体积之间的关系,公式为:
质量 (mg) = 浓度 (mM) x 体积 (mL) x 分子量 (g/mol)