S86115 |
Asenapine |
MedMol | 98% |
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- 产品描述: Asenapine (Org 5222), an atypical antipsychotic, is an antagonist of serotonin receptors (pKi: 8.4-10.5), adrenoceptors (pKi: 8.9-9.5), dopamine receptors (pKi: 8.9-9.4) and histamine receptors (pKi: 8.2-9.0). Asenapine can be used in the research of schizophrenia and bipolar disorder
- 靶点: 5-HT1A Receptor:8.6 (pKi);5-HT1B Receptor:8.4 (pKi);5-HT2A Receptor:10.2 (pKi);5-HT2B Receptor:9.8 (pKi);5-HT2C Receptor:10.5 (pKi);5-HT5 Receptor:8.8 (pKi);5-HT6 Receptor:9.6 (pKi);5-HT7 Receptor:9.9 (pKi);Alpha-2A adrenergic receptor:8.9 (pKi);α1-adrenergic receptor:8.9 (pKi);Alpha-2B adrenergic receptor:9.5 (pKi);Alpha-2C adrenergic receptor:8.9 (pKi);D1 Receptor:8.9 (pKi);D2 Receptor:8.9 (pKi);D3 Receptor:9.4 (pKi);D4 Receptor:9.0 (pKi);H1 Receptor:9.0 (pKi);H2 Receptor:8.2 (pKi)
- 体内研究: Asenapine (0.05-0.2 mg/kg; s.c.) induces a dose-dependent suppression of conditioned avoidance response (CAR) and does not induce catalepsy
- 参考文献:
1. M Shahid, et al. Asenapine: a novel psychopharmacologic agent with a unique human receptor signature. J Psychopharmacol. 2009 Jan;23(1):65-73. 2. Olivia Frånberg, et al. Asenapine, a novel psychopharmacologic agent: preclinical evidence for clinical effects in schizophrenia. Psychopharmacology (Berl). 2008 Feb;196(3):417-29.
- 溶解性: Soluble in DMSO
- 保存条件: -20℃
- 配置溶液浓度参考:
1mg 5mg 10mg 1 mM 3.499 ml 17.497 ml 34.993 ml 5 mM 0.7 ml 3.499 ml 6.999 ml 10 mM 0.35 ml 1.75 ml 3.499 ml 50 mM 0.07 ml 0.35 ml 0.7 ml
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本计算器可帮助您计算出特定溶液中溶质的质量、溶液浓度和体积之间的关系,公式为:
质量 (mg) = 浓度 (mM) x 体积 (mL) x 分子量 (g/mol)