| 货号 | 规格 | 价格 | 上海 | 北京 | 武汉 | 南京 | 购买数量 |
|---|---|---|---|---|---|---|---|
S80201-5mg |
99.7% | ￥270.00 | 10 | - | - | - |
|
S80201-10mg |
99.7% | ￥480.00 | 10 | - | - | - |
|
S80201-50mg |
99.7% | ￥1200.00 | >10 | - | - | - |
|
S80201-100mg |
99.7% | ￥2000.00 | >10 | - | - | - |
|
Azasetron (Y-25130) hydrochloride, a benzamide derivative, is a potent and selective 5-HT3 receptor antagonist. Azasetron is used in the study for Chemotherapy-induced nausea and vomiting (CINV)
| 产品描述： | Azasetron (Y-25130) hydrochloride, a benzamide derivative, is a potent and selective 5-HT3 receptor antagonist. Azasetron is used in the study for Chemotherapy-induced nausea and vomiting (CINV) | ||||||||||||||||||||
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| 靶点： | 5-HT3 Receptor：0.33 nM (IC50);5-HTReceptor | ||||||||||||||||||||
| 体内研究： | Azasetron could effectively penetrate through the skin and pass into the systemic circulation | ||||||||||||||||||||
| 参考文献： | 1. Sato, N., et al., Antagonistic activity of Y-25130 on 5-HT3 receptors. Jpn J Pharmacol, 1992. 59(4): p. 443-8. 2. Haga, K., et al., The effects of orally administered Y-25130, a selective serotonin3-receptor antagonist, on chemotherapeutic agent-induced emesis. Jpn J Pharmacol, 1993. 63(3): p. 377-83. | ||||||||||||||||||||
| 溶解性： | H2O : 20 mg/mL (51.78 mM; Need ultrasonic) DMSO : 2.22 mg/mL (5.75 mM; Need ultrasonic) | ||||||||||||||||||||
| 保存条件： | -20℃ | ||||||||||||||||||||
| 配置溶液浓度参考： |
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| 注意： | 部分产品我司仅能提供部分信息，我司不保证所提供信息的权威性，仅供客户参考交流研究之用。 |
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