H1 受体选择性抑制剂| 激动剂 | 拮抗剂;H1 receptor Selective Inhibitors | Agonists | Antagonists;;InformationPromethazine is a potenthistamine H1 receptorantagonist. Promethazine is a medication used in the management and treatment of allergic conditions, nausea and vomiting, motion sickness, and sedation. Promethazine exhibits antiparasitic properties.Targetshistamine H1 receptor
体内研究:
Promethazine (intraperitoneal injection; 2 mg/kg, 4 mg/kg, 6 mg/kg; once) is effective in reducing the writhing response.