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甲磺酸盐西地那非

    
10mM in DMSO

Sildenafil Mesylate

源叶(MedMol)
S57058 一键复制产品信息
1308285-21-3
C22H30N6O4S.xCH4O3S
474.58(free base)
7H-​Pyrazolo[4,​3-​d]​pyrimidin-​7-​one,5-​[2-​ethoxy-​5-​[(4-​methyl-​1-​piperazinyl)​sulfonyl]​phenyl]​-​1,​6-​dihydro-​1-​methyl-​3-​propyl-​,methanesulfonate (1:?)
货号 规格 价格 上海 北京 珠海 重庆 武汉 购买数量
S57058-1ml促销
10mM in DMSO

¥206.00 ¥185.00

9 - - - -
产品介绍 参考文献 质检证书(COA) 摩尔浓度计算器 相关产品
产品描述: PDE5 选择性抑制剂;PDE5 Selective Inhibitors;;InformationSildenafil Mesylate is a mesylate form of Sildenafil, an inhibitor ofPhosphodiesterase 5.TargetsPDE5In vivoChronic sildenafil treatment increases the detumescence phase in young and aged rats (p<0.05), although aged rats show a greater increase than young rats. Baseline cavernous PDE5 expression and activity are greater in aged vs young rats (p<0.05). After chronic sildenafil treatment cavernous PDE5 expression is increased in young (p<0.05) but not in aged rats. Chronic and acute sildenafil treatment similarly inhibits PDE5 activity in the penis of young and aged rats (p<0.05), coincident with its free plasma concentrations equivalent to clinically therapeutic ranges.
参考文献: 1. Haider M, et al. The Potential Role of Sildenafil in Cancer Management through EPR Augmentation. J Pers Med. 2021 Jun 21;11(6):585.
保存条件: -80℃(运输条件:冰袋低温运输)
配置溶液浓度参考:
1mg 5mg 10mg
1 mM 0 ml 0 ml 0 ml
5 mM 0 ml 0 ml 0 ml
10 mM 0 ml 0 ml 0 ml
50 mM 0 ml 0 ml 0 ml
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参考文献

质检证书(COA)

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摩尔浓度计算器

质量 (mg) = 浓度 (mM) x 体积 (mL) x 分子摩尔量 (g/mol)

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