| 货号 | 规格 | 价格 | 上海 | 北京 | 武汉 | 南京 | 购买数量 |
|---|---|---|---|---|---|---|---|
S80507-2mg |
99.7% | ￥180.00 | 5 | - | - | - |
|
S80507-5mg |
99.7% | ￥374.00 | 6 | - | - | - |
|
S80507-10mg |
99.7% | ￥586.50 | 6 | - | - | - |
|
S80507-25mg |
99.7% | ￥980.00 | 6 | - | - | - |
|
S80507-50mg |
99.7% | ￥1770.00 | 5 | - | - | - |
|
S80507-100mg |
≥98% | ￥2450.00 | 货期：2-3天 | - | - | - |
|
S80507-200mg |
≥98% | ￥4500.00 | 货期：2-3天 | - | - | - |
|
BRL-15572 dihydrochloride is a selective antagonist of h5-HT1D, displays high affinity for h5-HT1D receptors. BRL-15572 dihydrochloride could be useful pharmacological agents to characterise 5-HT1D receptor mediated responses
| 产品描述： | BRL-15572 dihydrochloride is a selective antagonist of h5-HT1D, displays high affinity for h5-HT1D receptors. BRL-15572 dihydrochloride could be useful pharmacological agents to characterise 5-HT1D receptor mediated responses | ||||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 靶点： | 5-HT1D Receptor;5-HTReceptor | ||||||||||||||||||||
| 体内研究： | BRL-15572 prevents (-)-epicatechin-induced antinociception in the formalin test. BRL-15572 (0.3-100.0 mg/kg; i.p.) is inactive and BRL-15572 (0.1-10 mg/kg; i.p.) has no effect on body temperature the guinea pig. | ||||||||||||||||||||
| 参考文献： | 1. Price GW, et, al. SB-216641 and BRL-15572--compounds to pharmacologically discriminate h5-HT1B and h5-HT1D receptors. Naunyn Schmiedebergs Arch Pharmacol. 1997 Sep; 356(3): 312-20. 2. Geovanna NQ, et, al. Antinociceptive effect of (-)-epicatechin in inflammatory and neuropathic pain in rats. Behav Pharmacol. 2018 Apr; 29(2 and 3-Spec Issue): 270-279. 3. Hagan JJ, et, al. Stimulation of 5-HT1B receptors causes hypothermia in the guinea pig. Eur J Pharmacol. 1997 Jul 23; 331(2-3): 169-74. | ||||||||||||||||||||
| 溶解性： | DMSO : 250 mg/mL (520.97 mM; Need ultrasonic) H2O : 2 mg/mL (4.17 mM; ultrasonic and warming and heat to 60°C) | ||||||||||||||||||||
| 保存条件： | -20℃ | ||||||||||||||||||||
| 配置溶液浓度参考： |
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| 注意： | 部分产品我司仅能提供部分信息，我司不保证所提供信息的权威性，仅供客户参考交流研究之用。 |
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