| 货号 | 规格 | 价格 | 上海 | 北京 | 珠海 | 重庆 | 武汉 | 购买数量 |
|---|---|---|---|---|---|---|---|---|
S80621-5mg买3赠1 |
98.75% | ￥528.00 |
1 | - | - | - | - |
|
S80621-10mg买3赠1 |
98.75% | ￥940.00 |
9 | - | - | - | - |
|
S80621-25mg买3赠1 |
98.75% | ￥1200.00 |
8 | - | - | - | - |
|
S80621-100mg买3赠1 |
≥98% | ￥1760.00 |
货期：2-3天 | - | - | - | - |
|
| 产品描述： | Regadenoson (CVT-3146) is a selective A2A adenosine receptor agonist and vasodilator that increases coronary blood flow, can be used in study of myocardial perfusion imaging. Regadenoson also increases the permeability of the blood-brain barrier (BBB) in rodents, can be used to study increased delivery of drugs to the human CNS | ||||||||||||||||||||
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| 靶点： | Adenosine Receptor;AdenosineReceptor | ||||||||||||||||||||
| 体内研究： | Regadenoson (0.1, 0.175, 0.25, 0.5, 1.0, 2.5, 5 µg/kg; p.i.v.; single) increases coronary blood flow (CBF) and decreases in mean coronary resistance in a dose-dependent manner, in awake dogs. Regadenoson (2.5 µg/kg; p.i.v.; single in 30 s) increases blood flow of coronary in awake dogs. Regadenoson (0.5 µg/kg; i.v.; single; 60 or 90 min after Temozolomide administration) promotes Temozolomide delivery to CNS of rats. | ||||||||||||||||||||
| 参考文献： | 1. Trochu JN, et al. Selective A2A adenosine receptor agonist as a coronary vasodilator in conscious dogs: potential for use in myocardial perfusion imaging. J Cardiovasc Pharmacol. 2003 Jan;41(1):132-9. 2. Jackson S, et al. The effect of regadenoson-induced transient disruption of the blood-brain barrier on temozolomide delivery to normal rat brain. J Neurooncol. 2016 Feb;126(3):433-9. | ||||||||||||||||||||
| 溶解性： | DMSO : 50 mg/mL (128.09 mM; Need ultrasonic) | ||||||||||||||||||||
| 保存条件： | -20℃ | ||||||||||||||||||||
| 配置溶液浓度参考： |
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| 注意： | 部分产品我司仅能提供部分信息，我司不保证所提供信息的权威性，仅供客户参考交流研究之用。 |
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