| 产品描述: | Zaurategrast ethyl ester sulfate (CDP323 sulfate), the ethyl ester prodrug of CT7758, is a α4β1/α4β7 integrin antagonist used for the treatment of inflammatory and autoimmune disorders |
| 靶点: |
α4β1/α4β7 integrin;Others |
| 参考文献: |
1. Chanteux H, et al. Cross-Species Differences in the Preclinical Pharmacokinetics of CT7758, an α4β1/α4β7 Integrin Antagonist. Drug Metab Dispos. 2015 Sep;43(9):1381-91. 2. Davenport RJ, et al. Alpha4-integrin antagonism--an effective approach for the treatment of inflammatory diseases? Drug Discov Today. 2007 Jul;12(13-14):569-76. |
| 保存条件: |
-20℃ |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
1.544 ml |
7.722 ml |
15.443 ml |
| 5 mM |
0.309 ml |
1.544 ml |
3.089 ml |
| 10 mM |
0.154 ml |
0.772 ml |
1.544 ml |
| 50 mM |
0.031 ml |
0.154 ml |
0.309 ml |
|
| 注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |