产品描述: c-Kit-IN-1 is a potent inhibitor of c-Kit and c-Met with IC50s of <200 nM. |
靶点:
IC50: <200 nM (c-Met), <200 nM (c-Kit), <2 μM (KDR), <10 μM (PDGFRα), <10 μM (PDGFRβ);c-Met/HGFR; c-Kit |
参考文献:
1. Daniel L. Flynn, et al. Cyclopropane amides and analogs exhibiting anti-cancer and anti-proliferative activities. WO 2010051373 A1 |
溶解性:
DMSO : ≥ 100 mg/mL (204.30 mM) |
保存条件:
-20℃ |
配置溶液浓度参考:
|
1mg |
5mg |
10mg |
1 mM |
2.043 ml |
10.215 ml |
20.43 ml |
5 mM |
0.409 ml |
2.043 ml |
4.086 ml |
10 mM |
0.204 ml |
1.022 ml |
2.043 ml |
50 mM |
0.041 ml |
0.204 ml |
0.409 ml |
|
注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |