| 货号 | 规格 | 价格 | 上海 | 北京 | 珠海 | 重庆 | 武汉 | 购买数量 |
|---|---|---|---|---|---|---|---|---|
S83760-5mg买3赠1 |
99.00% | ￥230.00 |
6 | - | - | - | - |
|
S83760-10mg买3赠1 |
99.00% | ￥400.00 |
6 | - | - | - | - |
|
S83760-25mg买3赠1 |
99.00% | ￥800.00 |
6 | - | - | - | - |
|
S83760-50mg |
99.00% | ￥1100.00 |
4 | - | - | - | - |
|
| 产品描述： | Namodenoson (CF-102) is a selective A3 adenosine receptor (A3AR) agonist (Ki=0.33 nM). Namodenoson displays 2500- and 1400-fold selectivity over A1 and A2A receptors respectively | ||||||||||||||||||||
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| 靶点： | Ki:0.33 nM (A3 adenosine receptor);AdenosineReceptor | ||||||||||||||||||||
| 体内研究： | Intravenous administration of 200 μg/kg Namodenoson (2-Cl-IB-MECA) resulted in a short-lasting hypotension, which was accompanied by a 50-100-fold increase in plasma histamine concentrations. Administration of a second dose of Namodenoson (2-Cl-IB-MECA) did not elicit any hemodynamic effects | ||||||||||||||||||||
| 参考文献： | 1. Van Schaick EA et al. Hemodynamic effects and histamine release elicited by the selective adenosine A3 receptor agonist 2-Cl-IB-MECA in conscious rats. Eur J Pharmacol. 1996 Jul 25;308(3):311-4. 2. Jacobson KA et al. Adenosine A3 receptors: novel ligands and paradoxical effects. Trends Pharmacol Sci. 1998 May;19(5):184-91. | ||||||||||||||||||||
| 溶解性： | DMSO : ≥ 31 mg/mL (56.91 mM) | ||||||||||||||||||||
| 保存条件： | 2-8℃ | ||||||||||||||||||||
| 配置溶液浓度参考： |
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| 注意： | 部分产品我司仅能提供部分信息，我司不保证所提供信息的权威性，仅供客户参考交流研究之用。 |
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