货号	规格	价格	上海	北京	珠海	重庆	武汉
S84292-5mg买3赠1	99.60%	￥65.00 S84292-5mg ￥65.00 现货（买3赠1）	1609 >10	-	-	-	-
S84292-10mg买3赠1	99.60%	￥100.00 S84292-10mg ￥100.00 现货（买3赠1）	803 >10	-	-	-	-
S84292-50mg买3赠1	99.60%	￥140.00 S84292-50mg ￥140.00 现货（买3赠1）	168 >10	-	-	-	-
S84292-250mg买3赠1	99.60%	￥340.00 S84292-250mg ￥340.00 现货（买3赠1）	38 >10	-	-	-	-

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产品描述：

Bilastine is a selective histamine H1 receptor antagonist used for treatment of allergic rhinoconjunctivitis and urticaria. Target: Histamine H1 Receptor Bilastine binds to histamine H1-receptors as indicated by its displacement of [3H]-pyrilamine from H1-receptors expressed in guinea-pig cerebellum and human embryonic kidney (HEK) cell lines. The studies conducted on guinea-pig smooth muscle demonstrated the capability of bilastine to antagonise H1-receptors. Bilastine is selective for histamine H1-receptors as shown in receptor-binding screening conducted to determine the binding capacity of bilastine to 30 different receptors [1]. Bilastine distribution has an apparent volume of distribution of 1.29 L/kg, and has an elimination half-life of 14.5 h and plasma protein binding of 84-90%

靶点：

Histamine Receptor;HistamineReceptor

体内研究：

In patients with allergic rhinoconjunctivitis, Bilastine is efficacious in all nasal symptoms including obstruction and in eye symptoms. In the fasting state, Bilastine is quickly absorbed, but the absorption is slowed when it is taken with food or fruit juice.

参考文献：

1.Wolthers OD.Bilastine: a new nonsedating oral H1 antihistamine for treatment of allergic rhinoconjunctivitis and urticaria.Biomed Res Int. 2013;2013:626837.

溶解性：

DMSO:10mM

保存条件：

2-8℃

配置溶液浓度参考：

	1mg	5mg	10mg
1 mM	2.157 ml	10.785 ml	21.57 ml
5 mM	0.431 ml	2.157 ml	4.314 ml
10 mM	0.216 ml	1.078 ml	2.157 ml
50 mM	0.043 ml	0.216 ml	0.431 ml

注意：

部分产品我司仅能提供部分信息，我司不保证所提供信息的权威性，仅供客户参考交流研究之用。

参考文献

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