| 货号 | 规格 | 价格 | 上海 | 北京 | 珠海 | 重庆 | 武汉 | 购买数量 |
|---|---|---|---|---|---|---|---|---|
S87592-5mg |
≥99% | ￥400.00 |
8 | - | - | - | - |
|
S87592-10mg |
≥99% | ￥680.00 |
4 | - | - | - | - |
|
S87592-25mg |
≥99% | ￥1350.00 |
4 | - | - | - | - |
|
S87592-50mg |
≥99% | ￥2390.00 |
2 | - | - | - | - |
|
S87592-100mg |
≥99% | ￥3590.00 |
2 | - | - | - | - |
|
| 产品描述： | Eltoprazine hydrochloride is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM, respectively). | ||||||||||||||||||||
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| 靶点： | 5-HT Receptor;5-HTReceptor | ||||||||||||||||||||
| 体内研究： | Eltoprazine hydrochloride exerts a dose-dependent decrease in aggressive behavior in resident-intruder tests with rats (ID50 = 0.24 mg/kg) | ||||||||||||||||||||
| 参考文献： | 1. Gravius A , Dekundy A , Vanaga A , et al. Further pharmacological characterization of eltoprazine: Focus on its anxiolytic, anorexic, and adverse-effect potential[J]. Acta neurobiologiae experimentalis, 2017, 77(1):77-85. 2. Boer S F D , Lesourd M , Mocaer E , et al. Selective Antiaggressive Effects of Alnespirone in Resident-Intruder Test Are Mediated via 5-Hydroxytryptamine1A Receptors: A Comparative Pharmacological Study with 8-Hydroxy-2-Dipropylaminotetralin, Ipsapirone, Buspirone, Eltoprazine, and WAY-100635[J]. Journal of Pharmacology & Experimental Therapeutics, 1999, 288(3):1125-1133. | ||||||||||||||||||||
| 溶解性： | Soluble in DMSO、H2O | ||||||||||||||||||||
| 保存条件： | 2-8℃ | ||||||||||||||||||||
| 配置溶液浓度参考： |
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| 注意： | 部分产品我司仅能提供部分信息，我司不保证所提供信息的权威性，仅供客户参考交流研究之用。 |
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