| 产品描述: | SR2640 (hydrochloride) 是一种有效且具有选择性与竞争性的 leukotriene D4/leukotriene E4 拮抗剂。SR2640 可用于研究白三烯在人类哮喘中的作用。 |
| 靶点: |
LTD4 and LTE4 |
| 体内研究: |
SR2640 inhibits the LTD 4-induced contractions of guinea-pig ileum in a concentration-dependent manner, with an IC50 of 3 nM. SR2640 (1 mg/kg; IV; single dosage) specifically prevents the contractile responses of guinea-pig ileum and trachea to LTD4 and LTE4. |
| 参考文献: |
1. Ahnfelt-Rønne I, Kirstein D, Kaergaard-Nielsen C. A novel leukotriene D4/E4 antagonist, SR2640 (2-[3-(2-quinolylmethoxy)phenylamino]benzoic acid). Eur J Pharmacol. 1988;155(1-2):117-128. |
| 溶解性: |
soluble in DMSO |
| 保存条件: |
-80℃(运输条件:冰袋低温运输) |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
2.458 ml |
12.289 ml |
24.578 ml |
| 5 mM |
0.492 ml |
2.458 ml |
4.916 ml |
| 10 mM |
0.246 ml |
1.229 ml |
2.458 ml |
| 50 mM |
0.049 ml |
0.246 ml |
0.492 ml |
|
| 注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |