PNU-282987 S enantiomer free base is an agonist of α7 nicotinic acetylcholine receptor (α7 nAChR)
靶点:
AChR
参考文献:
1. Bodnar A L , Cortes-Burgos L A , Cook K K , et al. Discovery and Structure?Activity Relationship of Quinuclidine Benzamides as Agonists of Nicotinic Acetylcholine Receptors[J]. Journal of Medicinal Chemistry, 2005, 48(4):905-908.