| 产品描述: | ATX inhibitor 1 is a potent ATX (IC50=1.23 nM, FS-3 and 2.18 nM, bis-pNPP) inhibitor. |
| 靶点: |
IC50: 1.23 nM (FS-3) and 2.18 nM (bis-pNPP) |
| 参考文献: |
1. Balupuri A, et al. Discovery and optimization of ATX inhibitors via modeling, synthesis and biological evaluation. Eur J Med Chem. 2018 Mar 25;148:397-409. |
| 溶解性: |
Soluble in DMSO |
| 保存条件: |
-80℃(运输条件:冰袋低温运输) |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
1.995 ml |
9.974 ml |
19.948 ml |
| 5 mM |
0.399 ml |
1.995 ml |
3.99 ml |
| 10 mM |
0.199 ml |
0.997 ml |
1.995 ml |
| 50 mM |
0.04 ml |
0.199 ml |
0.399 ml |
|
| 注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |