| 产品描述: | Val-Cit-PAB-MMAE is a?agent-linker conjugate for ADC. Val-Cit-PAB-MMAE contains the ADCs linker (peptide Val-Cit-PAB) and a potent tubulin inhibitor MMAE (HY-15162). MMAE?a potent?mitotic?inhibitor by inhibiting tubulin polymerization |
| 靶点: |
Auristatin |
| 参考文献: |
1. Okeley, et al. Intracellular Activation of SGN-35, a Potent Anti-CD30 Antibody-Drug Conjugate. Clinical Cancer Research (2010), 16(3), 888-897. |
| 溶解性: |
soluble in DMSO |
| 保存条件: |
-80℃(运输条件:冰袋低温运输) |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
0.89 ml |
4.451 ml |
8.901 ml |
| 5 mM |
0.178 ml |
0.89 ml |
1.78 ml |
| 10 mM |
0.089 ml |
0.445 ml |
0.89 ml |
| 50 mM |
0.018 ml |
0.089 ml |
0.178 ml |
|
| 注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |