| 产品描述: | NB-598 是一种有效的竞争性 squalene epoxidase (SE) 的抑制剂。NB-598 可抑制 cholesterol胆固醇 的生物合成 |
| 靶点: |
squalene epoxidase;cholesterol |
| 细胞实验: |
Cell lines: MIN6 cells Concentrations: 10 μM Incubation Time: 48 h Method: Cells were treated with indicated concentration of drug for 48 h. |
| 动物实验: |
Animal Models: Female CD rats Dosages: 5.1 mg/kg Administration: p.o. |
| 参考文献: |
1. Fuzhen Xia, et al. Endocrinology. 2008 Oct;149(10):5136-45. 2. Xia F, et al. Endocrinology. 2008 Oct;149(10):5136-45. 3. Horie M, et al. J Biol Chem. 1990 Oct 25;265(30):18075-8. |
| 溶解性: |
Soluble in DMSO、Ethanol |
| 保存条件: |
-80℃(运输条件:冰袋低温运输) |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
2.224 ml |
11.119 ml |
22.239 ml |
| 5 mM |
0.445 ml |
2.224 ml |
4.448 ml |
| 10 mM |
0.222 ml |
1.112 ml |
2.224 ml |
| 50 mM |
0.044 ml |
0.222 ml |
0.445 ml |
|
| 注意: |
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