| 产品描述: | SMCC-DM1 (DM1-SMCC) is a agent-linker conjugate composed of a potent microtubule-disrupting agent DM1 and a linker SMCC to make antibody agent conjugate (ADC) |
| 靶点: |
Maytansinoids |
| 体外研究: |
SMCC-DM1 抑制 HCC1954 和 MDA-MB-468 细胞增殖,IC50 分别为 17.2 和 49.9 nM |
| 参考文献: |
1. Shao S, et al. Site-specific and hydrophilic ADCs through disulfide-bridged linker and branched PEG. Bioorg Med Chem Lett. 2018 May 1;28(8):1363-1370. |
| 溶解性: |
Soluble in DMSO |
| 保存条件: |
-80℃(运输条件:冰袋低温运输) |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
0.932 ml |
4.662 ml |
9.323 ml |
| 5 mM |
0.186 ml |
0.932 ml |
1.865 ml |
| 10 mM |
0.093 ml |
0.466 ml |
0.932 ml |
| 50 mM |
0.019 ml |
0.093 ml |
0.186 ml |
|
| 注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |