| 体内研究: |
鞘内注射 TG003 (1-100 pM) 或 IC261 (0.1-1 nM) 可剂量依赖性地降低角叉菜胶或 CFA 引起的机械异常性疼痛和热痛觉过敏。 |
| 参考文献: |
1. Muraki M, et al. Manipulation of alternative splicing by a newly developed inhibitor of Clks. J Biol Chem. 2004 Jun 4;279(23):24246-54. 2. Marcel V, et al. Modulation of p53β and p53γ expression by regulating the alternative splicing of TP53 gene modifies cellular response. Cell Death Differ. 2014 Sep;21(9):1377-87. 3. Kurihara T, et al. Alleviation of behavioral hypersensitivity in mouse models of inflammatory pain with two structurally different casein kinase 1 (CK1) inhibitors. Mol Pain. 2014 Mar 10;10:17. |
| 保存条件: |
-80℃(运输条件:冰袋低温运输) |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
4.011 ml |
20.054 ml |
40.107 ml |
| 5 mM |
0.802 ml |
4.011 ml |
8.021 ml |
| 10 mM |
0.401 ml |
2.005 ml |
4.011 ml |
| 50 mM |
0.08 ml |
0.401 ml |
0.802 ml |
|
| 注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |