| 产品描述: | 胸苷酸合成酶抑制剂,也抑制二氢叶酸还原酶,GARFT和AICART;Thymidylate synthetase inhibitor, also inhibits dihydrofolate reductase, GARFT and AICART;Pemetrexed是抗叶酸和抗代谢剂,对TS,DHFR和GARFT的Ki分别为1.3 nM,7.2 nM和65 nM。;Pemetrexed is a novel antifolate and antimetabolite for TS, DHFR and GARFT with Ki of 1.3 nM, 7.2 nM and 65 nM, respectively. |
| 靶点: |
Ki: 1.3 nM (TS), 7.2 nM (DHFR), 65 nM (GARFT) |
| 保存条件: |
-80℃(运输条件:冰袋低温运输) |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
2.34 ml |
11.698 ml |
23.397 ml |
| 5 mM |
0.468 ml |
2.34 ml |
4.679 ml |
| 10 mM |
0.234 ml |
1.17 ml |
2.34 ml |
| 50 mM |
0.047 ml |
0.234 ml |
0.468 ml |
|
| 注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |