| 产品描述: | AI-10-49 is a selective inhibitor of the binding of CBFβ-SMMHC to RUNX1 with IC50 of 260 nM. |
| 体内研究: |
AI-10-49 (200 mg/kg;每天) 延缓小鼠白血病的进展。 |
| 参考文献: |
1. Anuradha Illendula, et al. Chemical biology. A small-molecule inhibitor of the aberrant transcription factor CBFβ-SMMHC delays leukemia in mice. Science. 2015 Feb 13;347(6223):779-84. |
| 保存条件: |
-80℃(运输条件:冰袋低温运输) |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
1.514 ml |
7.57 ml |
15.14 ml |
| 5 mM |
0.303 ml |
1.514 ml |
3.028 ml |
| 10 mM |
0.151 ml |
0.757 ml |
1.514 ml |
| 50 mM |
0.03 ml |
0.151 ml |
0.303 ml |
|
| 注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |