| 产品描述: | 抗菌和抗寄生虫剂;Antibacterial and antiparasitic agent;Closantel是革兰氏阳性的抗菌活性抑制剂,抑制KinA/Spo0F系统,IC50为3.8 μM。;Closantel is a gram positive antibacterial activity inhibitor, inhibiting the KinA/Spo0F system with IC50 of 3.8 μM.Potentially useful for studying P-glycoprotein interactions in vitro. |
| 参考文献: |
1. Amanda L Garner, et al. Design, synthesis, and biological activities of closantel analogues: structural promiscuity and its impact on Onchocerca volvulus. J Med Chem. 2011 Jun 9;54(11):3963-72. 2. Amanda L Garner, et al. Design, synthesis, and biological activities of closantel analogues: structural promiscuity and its impact on Onchocerca volvulus. J Med Chem. 2011 Jun 9;54(11):3963-72. |
| 保存条件: |
-80℃(运输条件:冰袋低温运输) |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
1.508 ml |
7.541 ml |
15.081 ml |
| 5 mM |
0.302 ml |
1.508 ml |
3.016 ml |
| 10 mM |
0.151 ml |
0.754 ml |
1.508 ml |
| 50 mM |
0.03 ml |
0.151 ml |
0.302 ml |
|
| 注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |