| 产品描述: | 强大的选择性细胞渗透性EZH2甲基转移酶抑制剂;Potent, selective cell-permeable EZH2 methyltransferase inhibitor;UNC1999是口服生物相容性的EZH2和EZH1抑制剂,IC50分别为2 nM和45 nM。;UNC1999 is a potent, orally bioavailable and selective inhibitor of EZH2 and EZH1 with IC50 of 2 nM and 45 nM in cell-free assays, respectively, showing >1000-fold selectivity over a broad range of epigenetic and non-epigenetic targets. |