| 靶点: |
IC50: 5 μM (ACE) |
| 体内研究: |
Ile-Pro-Pro (IPP; 30 mg/kg per day; 0.3 g/L) attenuates arterial dysfunction in L-NAME-treated rats Ile-Pro-Pro decreases blood pressure in spontaneously hypertensive rats (SHR) . Ile-Pro-Pro attenuates the development of atherosclerosis in apolipoprotein E-deficient (apoE(-/-)) mice. |
| 参考文献: |
1. Nonaka A, et al. The milk-derived peptides Val-Pro-Pro and Ile-Pro-Pro attenuate arterial dysfunction in L-NAME-treated rats. Hypertens Res. 2014 Aug;37(8):703-7. 2. Nakamura Y, et al. Purification and characterization of angiotensin I-converting enzyme inhibitors from sour milk. J Dairy Sci. 1995 Apr;78(4):777-83. |
| 保存条件: |
-80℃,避光,干燥(运输条件:冰袋低温运输) |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
2.763 ml |
13.817 ml |
27.635 ml |
| 5 mM |
0.553 ml |
2.763 ml |
5.527 ml |
| 10 mM |
0.276 ml |
1.382 ml |
2.763 ml |
| 50 mM |
0.055 ml |
0.276 ml |
0.553 ml |
|
| 注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |