| 靶点: |
IC50: 25 nM (Rat ACAT), 44 nM (Rabbit ACAT) |
| 体内研究: |
RP 70676 (10 mg/kg, p.o.) is well absorbed with plasma levels in NZW rabbits. |
| 参考文献: |
1. M.J. Ashton, et al. RP 70676: A potent systematically available inhibitor of acyl-CoA:cholesterol O-acyl transferase (ACAT). Bioorganic & Medicinal Chemistry Letters Volume 2, Issue 5, 1992, Pages 375-380. |
| 保存条件: |
-80℃(运输条件:冰袋低温运输) |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
2.4 ml |
12.002 ml |
24.005 ml |
| 5 mM |
0.48 ml |
2.4 ml |
4.801 ml |
| 10 mM |
0.24 ml |
1.2 ml |
2.4 ml |
| 50 mM |
0.048 ml |
0.24 ml |
0.48 ml |
|
| 注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |