| 靶点: |
Mps1 50 nM (IC50) |
| 体内研究: |
Mps1-IN-3 (2 mg/kg, i.v.) sensitizes glioblastoma cells in murine tumor models, with prolonged survival and no toxicity. |
| 参考文献: |
1. Tannous BA, et al. Effects of the selective MPS1 inhibitor MPS1-IN-3 on glioblastoma sensitivity to antimitotic drugs. J Natl Cancer Inst. 2013 Sep 4;105(17):1322-31. |
| 保存条件: |
-80℃(运输条件:冰袋低温运输) |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
1.86 ml |
9.3 ml |
18.6 ml |
| 5 mM |
0.372 ml |
1.86 ml |
3.72 ml |
| 10 mM |
0.186 ml |
0.93 ml |
1.86 ml |
| 50 mM |
0.037 ml |
0.186 ml |
0.372 ml |
|
| 注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |