IL 受体抑制剂;IL Receptor Inhibitors;产品介绍:IRAK4-IN-2 是一种可逆性激酶抑制剂,在TLR和IL-1R信号级联反应中,调节IRAK4的功能。;InformationIRAK4-IN-2 IRAK4-IN-2 is a reversible kinase inhibitor that modulates IRAK4 function in both the toll-like receptor (TLR) and interleukin 1 receptor (IL-1R) signaling cascades.TargetsIRAK4
体内研究:
IRAK4-IN-7 具有抗癌和抗炎活性,可用于癌症和炎症性疾病的处理。
参考文献:
1. Venkateshwar Rao GUMMADI, et al. Bicyclic heterocyclyl derivatives as irak4 inhibitors. WO2015104688A1.