| 靶点: |
Sodium Channel |
| 体内研究: |
给予 100 mg 和 150 mg Eniporide hydrochloride 导致梗塞面积变小,尤其是在血管成形术组。 |
| 参考文献: |
1. Klass O, et al. Effect of the Na+/H+ exchange inhibitor eniporide on cardiac performance and myocardial high energy phosphates in pigs subjected to cardioplegic arrest. Ann Thorac Surg. 2004 Feb;77(2):658-63. 2. Zeymer U, et al. The Na(+)/H(+) exchange inhibitor eniporide as an adjunct to early reperfusion therapy for acute myocardial infarction. Results of the evaluation of the safety and cardioprotective effects of eniporide in acute myocardial infarction (ESCAMI) trial. J Am Coll Cardiol. 2001 Nov 15;38(6):1644-50. |
| 保存条件: |
-80℃,干燥(运输条件:冰袋低温运输) |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
2.802 ml |
14.012 ml |
28.025 ml |
| 5 mM |
0.56 ml |
2.802 ml |
5.605 ml |
| 10 mM |
0.28 ml |
1.401 ml |
2.802 ml |
| 50 mM |
0.056 ml |
0.28 ml |
0.56 ml |
|
| 注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |