| 产品描述: | ICA-069673是KCNQ2/Q3钾通道激活剂,IC50值为0.69 μM。参考MCE |
| 靶点: |
IC50: 0.69 μM (KV7.2/7.3), 14.3 μM (KV7.3/7.5) |
| 参考文献: |
1. Provence A, et al. The Novel KV7.2/KV7.3 Channel Opener ICA-069673 Reveals Subtype-Specific Functional Roles in Guinea Pig Detrusor Smooth Muscle Excitability and Contractility. J Pharmacol Exp Ther. 2015 Sep;354(3):290-301. |
| 保存条件: |
-80℃(运输条件:冰袋低温运输) |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
3.709 ml |
18.544 ml |
37.088 ml |
| 5 mM |
0.742 ml |
3.709 ml |
7.418 ml |
| 10 mM |
0.371 ml |
1.854 ml |
3.709 ml |
| 50 mM |
0.074 ml |
0.371 ml |
0.742 ml |
|
| 注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |