| 体内研究: |
R243 (0.1-1 mg/kg;腹膜内注射;一次;雄性瑞士小鼠) 治疗以剂量依赖性方式抑制 CCL1 引起的镇痛作用。 |
| 参考文献: |
1. Tomoyuki Oshio, et al. Chemokine Receptor CCR8 Is Required for Lipopolysaccharide-Triggered Cytokine Production in Mouse Peritoneal Macrophages. PLoS One. 2014 Apr 8;9(4):e94445. 2. Mario García-Domínguez, et al. The Systemic Administration of the Chemokine CCL1 Evokes Thermal Analgesia in Mice Through the Activation of the Endocannabinoid System. Cell Mol Neurobiol. 2019 Nov;39(8):1115-1124. |
| 保存条件: |
-80℃(运输条件:冰袋低温运输) |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
2.798 ml |
13.988 ml |
27.977 ml |
| 5 mM |
0.56 ml |
2.798 ml |
5.595 ml |
| 10 mM |
0.28 ml |
1.399 ml |
2.798 ml |
| 50 mM |
0.056 ml |
0.28 ml |
0.56 ml |
|
| 注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |