DB07268是JNK1抑制剂,IC50为9 nM。;DB07268 is a potent and selective JNK1 inhibitor with an IC50 value of 9 nM.
参考文献:
1. Liu M, et al. Discovery of a new class of 4-anilinopyrimidines as potent c-Jun N-terminal kinase inhibitors: Synthesis and SAR studies. Bioorg Med Chem Lett. 2007 Feb 1;17(3):668-72.