| 体内研究: |
nor-NOHA monoacetate (100 mg/kg,静脉注射,一次) 可显著减少雄性 Sprague-Dawley 大鼠的梗塞面积。 nor-NOHA monoacetate (100 mg/kg,静脉注射,一次) 会增加雄性 Sprague-Dawley 大鼠的血浆中瓜氨酸和亚硝酸盐水平,并降低血浆中鸟氨酸水平。 |
| 参考文献: |
1. Ng KP, et al. The arginase inhibitor Nω-hydroxy-nor-arginine (nor-NOHA) induces apoptosis in leukemic cells specifically under hypoxic conditions but CRISPR/Cas9 excludes arginase 2 (ARG2) as the functional target. PLoS One. 2018 Oct 11;13(10):e0205254. 2. Jung C, et al. Arginase inhibition mediates cardioprotection during ischaemia-reperfusion. Cardiovasc Res. 2010 Jan 1;85(1):147-54. |
| 保存条件: |
2-8°C,干燥,密封 |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
4.233 ml |
21.166 ml |
42.332 ml |
| 5 mM |
0.847 ml |
4.233 ml |
8.466 ml |
| 10 mM |
0.423 ml |
2.117 ml |
4.233 ml |
| 50 mM |
0.085 ml |
0.423 ml |
0.847 ml |
|
| 注意: |
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