| 产品描述: | Lysipressin (Lysine vasopressin) is antidiuretic hormone that have been found in pigs and some marsupial families. Lysipressin induces contraction of the rabbit urinary bladder smooth muscle, activate adenylate-cyclase |
| 靶点: |
Adenylate Cyclase |
| 体内研究: |
Lysipressin (150-500 ng,ICV) 在大鼠中表现出抗伤害活性,增加甩尾反应延迟。 Lysipressin (0.1-100 mu/kg,静脉注射) 可升高狗的血压并降低心率。 Lysipressin (0.01-10 mu/kg,脑池内注射) 可引起与剂量相关的血压下降,但不改变狗的心率。 |
| 参考文献: |
1. Gorbulev V et al. Molecular cloning and functional characterization of V2 [8-lysine] vasopressin and oxytocin receptors from a pig kidney cell line. Eur J Biochem. 1993 Jul 1;215(1):1-7. 2. Crankshaw D et al. [Arg8]vasopressin-induced contractions of rabbit urinary bladder smooth muscle.Eur J Pharmacol. 1989 Dec 7;173(2-3):183-8. |
| 溶解性: |
Soluble in H2O |
| 保存条件: |
-80℃(运输条件:冰袋低温运输) |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
0.947 ml |
4.734 ml |
9.468 ml |
| 5 mM |
0.189 ml |
0.947 ml |
1.894 ml |
| 10 mM |
0.095 ml |
0.473 ml |
0.947 ml |
| 50 mM |
0.019 ml |
0.095 ml |
0.189 ml |
|
| 注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |