| 产品描述: | METTL1-WDR4-IN-2, an adenosine derivative, is a selective methyltransferase Like 1 (METTL1)-WDR4 inhibitor with an IC50 of 41 μM. METTL1-WDR4-IN-2 shows selectivity against METTL3-14 (IC50 of 958 μM) and METTL16 (IC50 of 208 μM). METTL1-WDR4-IN-2 can be used for the study of cancer. |
| 体外研究: |
METTL1-WDR4-IN-2 (compound 6) 在热位移分析中能够稳定 METTL1 和 METTL1-WDR4。 |
| 保存条件: |
-20°C |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
1.963 ml |
9.813 ml |
19.626 ml |
| 5 mM |
0.393 ml |
1.963 ml |
3.925 ml |
| 10 mM |
0.196 ml |
0.981 ml |
1.963 ml |
| 50 mM |
0.039 ml |
0.196 ml |
0.393 ml |
|
| 注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |