Oxidized ATP (oATP) trisodium salt is a broad-spectrum P2 receptor inhibitor. Oxidized ATP trisodium salt irreversibly antagonizes P2X7R activation. Oxidized ATP trisodium salt inhibits c-reactive protein (CRP)-induced NLRP3 inflammasome activation. Oxidized ATP trisodium salt can be used for research of atherosclerosis.
体外研究:
Oxidized ATP trisodium salt (100 μM,1 小时) 抑制 HUVEC 中 CRP (20 μg/mL,24 小时) 诱导的 caspase-1 激活和 IL-1β 成熟。