| 靶点: |
Na+channel |
| 体内研究: |
术前用 Ralfinamide (30 mg/kg、60 mg/kg;口服;每天两次;42 天) 或 Ralfinamide (80 mg/kg;口服;每天两次;7 天) 处理可抑制神经性疼痛。 |
| 参考文献: |
1. Zhang SH, et al. Ralfinamide administered orally before hindpaw neurectomy or postoperatively provided long-lasting suppression of spontaneous neuropathic pain-related behavior in the rat. Pain. 2008 Oct 15;139(2):293-305. 2. Liang X, et al. Effects of ralfinamide in models of nerve injury and chemotherapy-induced neuropathic pain. Eur J Pharmacol. 2018 Mar 15;823:27-34. |
| 保存条件: |
-80℃(运输条件:冰袋低温运输) |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
3.308 ml |
16.538 ml |
33.075 ml |
| 5 mM |
0.662 ml |
3.308 ml |
6.615 ml |
| 10 mM |
0.331 ml |
1.654 ml |
3.308 ml |
| 50 mM |
0.066 ml |
0.331 ml |
0.662 ml |
|
| 注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |