| 体内研究: |
TC I-15 (10 μg; 静脉注射; 每隔一天; 三周) 在小鼠中抑制了由 CAFs EVs 促进的肺转移。 |
| 参考文献: |
1. Emma J. Hunter, Selectivity of the collagen-binding integrin inhibitors, TC-I-15 and obtustatin. Toxicol Appl Pharmacol. 2021 Oct 1;428:115669. 2. Jing Kong, et al. Extracellular vesicles of carcinoma-associated fibroblasts creates a pre-metastatic niche in the lung through activating fibroblasts. Mol Cancer. 2019 Dec 3;18(1):175. |
| 保存条件: |
-80℃(运输条件:冰袋低温运输) |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
1.921 ml |
9.604 ml |
19.208 ml |
| 5 mM |
0.384 ml |
1.921 ml |
3.842 ml |
| 10 mM |
0.192 ml |
0.96 ml |
1.921 ml |
| 50 mM |
0.038 ml |
0.192 ml |
0.384 ml |
|
| 注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |