| 产品描述: | AChE-IN-26 (compound 4a) 是 AChE (acetylcholinesterase) 的抑制剂,IC50 值为 0.42 μM。AChE-IN-26 可用于阿尔兹海默症的研究。 |
| 靶点: |
IC50: 0.42 μM (AChE) |
| 体外研究: |
AChE-IN-26 (1 and 10 μM;20 min) shows an in-vitro inhibition to AChE of 91.45%, and inhibits AChE with an IC50 value of 0.42 μM. |
| 参考文献: |
1.Abdullaha M, et al. Discovery of methoxy-naphthyl linked N-(1-benzylpiperidine) benzamide as a blood-brain permeable dual inhibitor of acetylcholinesterase and butyrylcholinesterase. Eur J Med Chem. 2020 Dec 1;207:112761. |
| 保存条件: |
-80℃(运输条件:冰袋低温运输) |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
2.329 ml |
11.647 ml |
23.293 ml |
| 5 mM |
0.466 ml |
2.329 ml |
4.659 ml |
| 10 mM |
0.233 ml |
1.165 ml |
2.329 ml |
| 50 mM |
0.047 ml |
0.233 ml |
0.466 ml |
|
| 注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |