| 体内研究: |
Chlorothymol 在各种小鼠癫痫模型中发挥抗惊厥功效,包括 6-Hz 32-mA (ED50 = 18.0 mg/kg,保护指数 [PI] = 8.4、6-Hz 44-mA (ED50 = 66.2 mg/kg,PI = 2.3)。 |
| 参考文献: |
1. Alistair Jones, et al. A multiorganism pipeline for antiseizure drug discovery: Identification of chlorothymol as a novel γ-aminobutyric acidergic anticonvulsant. Epilepsia. 2020 Oct;61(10):2106-2118. 2. Kim BC, et al. 4-Chloro-2-Isopropyl-5-Methylphenol Exhibits Antimicrobial and Adjuvant Activity against Methicillin-Resistant Staphylococcus aureus. J Microbiol Biotechnol. 2022 Jun 28;32(6):730-739. |
| 保存条件: |
-80℃(运输条件:冰袋低温运输) |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
5.415 ml |
27.077 ml |
54.154 ml |
| 5 mM |
1.083 ml |
5.415 ml |
10.831 ml |
| 10 mM |
0.542 ml |
2.708 ml |
5.415 ml |
| 50 mM |
0.108 ml |
0.542 ml |
1.083 ml |
|
| 注意: |
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