IC50: 3.3 μM (trypanothione reductase) and 64.8 μM (glutathione reductase);EC50: 1 μM (T. brucei)
参考文献:
1. Martyn DC, et al. High-throughput screening affords novel and selective trypanothione reductase inhibitors with anti-trypanosomal activity. Bioorg Med Chem Lett. 2007 Mar 1;17(5):1280-3.