| 产品描述: | Cathepsin Inhibitor 2 是一种有效的 Cathepsin S 抑制剂,Ki 值 <20 nM。详细信息请参考专利文献 WO2009123623A1 中的段落 0229。 |
| 靶点: |
Ki: <20 nM (Cathepsin S) |
| 体内研究: |
Cathepsin Inhibitor 2 (Please refer to paragraph 0229 for detailed information) potently inhibits Cathepsin S, Cathepsin F, Cathepsin L, and Cathepsin B with Kis of <20 nM, 21-500 nM, 21-500 nM, and 21-500 nM, respectively[1]. |
| 参考文献: |
1. LINK, John, O, et al. DI-FLUORO CONTAINING COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS. WO2009123623A1. |
| 保存条件: |
-80°C 6个月;-20°C 1个月 |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
2.373 ml |
11.866 ml |
23.732 ml |
| 5 mM |
0.475 ml |
2.373 ml |
4.746 ml |
| 10 mM |
0.237 ml |
1.187 ml |
2.373 ml |
| 50 mM |
0.047 ml |
0.237 ml |
0.475 ml |
|
| 注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |