| 产品描述: | KP-302 (Compound 23) is a selective inhibitor of protein arginine deaminase PAD2 with a Ki of 60 μM. KP-302 also reverses physical disability in the EAE mouse model of multiple sclerosis (MS) and eliminates T cell infiltration in the brain. KP-302 can be studied in research as a disease-modifying agent for MS. |
| 体外研究: |
KP-302 (50 mg/kg,腹腔注射,每日一次) 对小鼠模型中的炎症脱髓鞘具有非常显著的保护作用[2]。 |
| 体内研究: |
KP-302 (50 mg/kg,腹腔注射,每日一次) 对小鼠模型中的炎症脱髓鞘具有非常显著的保护作用。 |
| 保存条件: |
-80°C 6个月;-20°C 1个月 |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
2.737 ml |
13.683 ml |
27.365 ml |
| 5 mM |
0.547 ml |
2.737 ml |
5.473 ml |
| 10 mM |
0.274 ml |
1.368 ml |
2.737 ml |
| 50 mM |
0.055 ml |
0.274 ml |
0.547 ml |
|
| 注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |