| 产品描述: | 5-HT2C agonist-3 ((+)-19) is a selective 5-HT2C agonist (EC50: 24 nM, Ki: 78 nM). 5-HT2C agonist-3 has antipsychotic drug-like activity. 5-HT2C agonist-3 blocks Amphetamine-induced hyperactivity. |
| 靶点: |
5-HT2C Receptor |
| 参考文献: |
1. Guiping Zhang, et al. Discovery of N-Substituted (2-Phenylcyclopropyl)methylamines as Functionally Selective Serotonin 2C Receptor Agonists for Potential Use as Antipsychotic Medications. J. Med. Chem. 2017, 60, 14, 6273–6288. |
| 保存条件: |
-80°C 12个月; -20°C 6个月, 干燥 |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
2.842 ml |
14.211 ml |
28.422 ml |
| 5 mM |
0.568 ml |
2.842 ml |
5.684 ml |
| 10 mM |
0.284 ml |
1.421 ml |
2.842 ml |
| 50 mM |
0.057 ml |
0.284 ml |
0.568 ml |
|
| 注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |