| 产品描述: | VU6010572 is a potent and selective mGlu3 negative allosteric modulator with IC50 of 245 nM. VU6010572 is highly CNS penetrant. |
| 靶点: |
mGluR3:245 nM (IC50) |
| 体外研究: |
VU6010572 (3 mg/kg; i.p.) shows robust efficacy[1]. VU6010572 (3 mg/kg; i.p.; 45 minutes) produces lasting anxiolytic-like behavioral effects[2]. |
| 保存条件: |
-80°C 6个月; -20°C 1个月,避光,氮气保存 |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
2.947 ml |
14.734 ml |
29.467 ml |
| 5 mM |
0.589 ml |
2.947 ml |
5.893 ml |
| 10 mM |
0.295 ml |
1.473 ml |
2.947 ml |
| 50 mM |
0.059 ml |
0.295 ml |
0.589 ml |
|
| 注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |