| 产品描述: | TRPV2-selective blocker 1 (compound IV2-1) is a selective TRPV2 channel blocker with an IC50 of 6.3 μM. TRPV2-selective blocker 1 does not affect TRPV1, TRPV3 or TRPV4 channels. TRPV2-selective blocker 1 also inhibits TRPV2-mediated Ca2+ influx in macrophages, and inhibits macrophage phagocytosis. |
| 靶点: |
TRPV2:6.3 μM (IC50) |
| 保存条件: |
-80°C 6个月; -20°C 1个月,避光,氮气保存 |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
3.592 ml |
17.958 ml |
35.916 ml |
| 5 mM |
0.718 ml |
3.592 ml |
7.183 ml |
| 10 mM |
0.359 ml |
1.796 ml |
3.592 ml |
| 50 mM |
0.072 ml |
0.359 ml |
0.718 ml |
|
| 注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |