| 产品描述: | (S)-GSK852 is a diastereomer of GSK852 . GSK852 is a BET inhibitor targeting BD2 (pIC50=7.9). |
| 参考文献: |
1. Lucas SCC, et al. Optimization of a Series of 2,3-Dihydrobenzofurans as Highly Potent, Second Bromodomain (BD2)-Selective, Bromo and Extra-Terminal Domain (BET) Inhibitors. J Med Chem. 2021 Aug 12;64(15):10711-10741. |
| 保存条件: |
-80°C 6个月;-20°C 1个月 |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
2.46 ml |
12.301 ml |
24.602 ml |
| 5 mM |
0.492 ml |
2.46 ml |
4.92 ml |
| 10 mM |
0.246 ml |
1.23 ml |
2.46 ml |
| 50 mM |
0.049 ml |
0.246 ml |
0.492 ml |
|
| 注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |