| 产品描述: | PROTAC BRD4 Degrader-12 (compound 9c) is a PROTAC connected by ligands for von Hippel-Lindau and BRD4. PROTAC BRD4 Degrader-12 can be conjugated with STEAP1 and CLL1 antibodies to degrade the BRD4 protein in PC3 prostate cancer cells, with a DC50 of 0.39 nM and 0.24 nM, respectively. |
| 保存条件: |
-80°C 6个月; -20°C 1个月,干燥,避光 |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
0.765 ml |
3.827 ml |
7.654 ml |
| 5 mM |
0.153 ml |
0.765 ml |
1.531 ml |
| 10 mM |
0.077 ml |
0.383 ml |
0.765 ml |
| 50 mM |
0.015 ml |
0.077 ml |
0.153 ml |
|
| 注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |