| 产品描述: | Pociredir (FTX-6058) is a potent and orally active inhibitor of Embryonic Ectoderm Development (EED). Pociredir can induce HbF protein expression in cell and murine models. Pociredir can be used for the research of select hemoglobinopathies, including sickle cell disease and β-thalassemia. |
| 体内研究: |
FTX-6058 通过与 EED 结合抑制 PRC2,从而在细胞和小鼠模型中诱导 HbF 蛋白的强表达。 |
| 参考文献: |
1. Boerner LK. Virtual meeting delivers first time drug structures. April 12, 2021. |
| 保存条件: |
-80°C 6个月;-20°C 1个月 |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
2.479 ml |
12.394 ml |
24.789 ml |
| 5 mM |
0.496 ml |
2.479 ml |
4.958 ml |
| 10 mM |
0.248 ml |
1.239 ml |
2.479 ml |
| 50 mM |
0.05 ml |
0.248 ml |
0.496 ml |
|
| 注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |