| 产品描述: | (1S,9R)-Exatecan mesylate ((1S,9R)-DX8951f) is an isomer of Exatecan mesylate . Exatecan mesylate (DX8951f) is an inhibitor of DNA topoisomerase I with an IC50 of 2.2 μM (0.975 μg/mL) and can be used in cancer research. |
| 靶点: |
Camptothecins |
| 参考文献: |
1. Mitsui I, et al. A new water-soluble camptothecin derivative, DX-8951f, exhibits potent antitumor activity against human tumors in vitro and in vivo. Jpn J Cancer Res. 1995 Aug;86(8):776-82. |
| 保存条件: |
-80°C 12个月; -20°C 6个月,干燥, 避光 |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
1.881 ml |
9.406 ml |
18.813 ml |
| 5 mM |
0.376 ml |
1.881 ml |
3.763 ml |
| 10 mM |
0.188 ml |
0.941 ml |
1.881 ml |
| 50 mM |
0.038 ml |
0.188 ml |
0.376 ml |
|
| 注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |