| 产品描述: | AMA-37, an Arylmorpholine analog, is ATP-competitive DNA-PK inhibitor, with IC50 values of 0.27 μM (DNA-PK), 32 μM (p110α), 3.7 μM (p110β), and 22 μM (p110γ), respectively. |
| 体内研究: |
AMA-37 inhbits PI3K poorly. AMA-37 (20 μM) reduces the ability of UCN-01, isogranulatimide, and debromohymenialdesine, but not caffeine, to overcome G2 arrest (ρ < 0.05). Inhibition of DNA-PK with AMA37 leads to radiosensitization. |
| 保存条件: |
-80°C 6个月;-20°C 1个月 |
| 配置溶液浓度参考: |
|
1mg |
5mg |
10mg |
| 1 mM |
3.53 ml |
17.648 ml |
35.296 ml |
| 5 mM |
0.706 ml |
3.53 ml |
7.059 ml |
| 10 mM |
0.353 ml |
1.765 ml |
3.53 ml |
| 50 mM |
0.071 ml |
0.353 ml |
0.706 ml |
|
| 注意: |
部分产品我司仅能提供部分信息,我司不保证所提供信息的权威性,仅供客户参考交流研究之用。 |